BPR5K230 is a dual inhibitor for the receptor tyrosine kinase MER and AXL, with IC50 of 4.1 nM and 9.2 nM. BPR5K230 inhibits the proliferation of Ba/F3-MER with IC50 of 5 nM. BPR5K230 exhibits good pharmacokinetic characteristics in mice, exhibits anti-inflammatory and antitumor against 4T1, MDA-MB-231, MC38 and Hepa1 6 in mouse models[1].
Molecular Weight:
655.68
Purity:
99.82
CAS Number:
[3029897-97-7]
Formula:
C37H30FN7O4
Target:
TAM Receptor
Application Notes:
MCE Product type: Reference compound
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