I-BET787 is a orally active BET bromine domain inhibitor with pIC50s of 7.1 and 5.9 for BRD4 BD1 and BRD4 BD2, respectively. I-BET787 has anti-inflammatory activity in mice[1].
Molecular Weight:
321.80
Purity:
99.88
CAS Number:
[2201082-98-4]
Formula:
C16H20ClN3O2
Target:
Epigenetic Reader Domain
Application Notes:
MCE Product type: Reference compound
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