CP-609754 (LNK-754) is a potent and reversible farnesyltransferase inhibitor with potential anticancer activity.The IC50 for inhibiting farnesylation of recombinant human H-Ras is 0.57 ng/mL and recombinant K-Ras is 46 ng/mL[1]. CP-609754 is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.
Molecular Weight:
479.96
Purity:
99.21
CAS Number:
[1190094-64-4]
Formula:
C29H22ClN3O2
Target:
Farnesyl Transferase
Application Notes:
MCE Product type: Reference compound
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