CysLT1 receptor antagonist-1 (Compound 4) is an antagonist for cysteinyl leukotriene receptor 1 (CysLT1R) with an IC50 of 3.9 µM. CysLT1 receptor antagonist-1 exhibits weak agonist activity against G-protein-coupled bile acid receptor 1 (GPBAR1) with an efficact of 23% at 10 µM. CysLT1 receptor antagonist-1 can be used for asthma and allergic diseases researchs[1].
Molecular Weight:
293.32
CAS Number:
[119515-00-3]
Formula:
C18H15NO3
Target:
Leukotriene Receptor
Application Notes:
MCE Product type: Reference compound
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