VUF14480 is a partial agonist of histamine H4 (hH4) receptor-mediated G protein signalling and beta-arrestin2 recruitment. VUF14480 binds covalently to hH4 receptor (pKi: 6.3 for hH4-WT receptor). VUF14480 partially induces hH4 receptor-mediated G protein activation and beta-arrestin2 recruitment. VUF14480 can be used in the research of inflammatory diseases[1].
Molecular Weight:
280.38
CAS Number:
[1605304-31-1]
Formula:
C17H20N4
Target:
Histamine Receptor
Application Notes:
MCE Product type: Reference compound
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