CID 16020046 is a potent and selective GPR55 antagonist and inhibits GPR55 constitutive activity with an IC50 of 0.15 µM. CID 16020046 inhibits GPR55-mediated Ca2+ signaling and GPR55-mediated ERK1/2 phosphorylation. CID 16020046 reduces wound healing in endothelial cells and is involved in the regulation of platelet function[1].
Molecular Weight:
425.44
Purity:
99.81
CAS Number:
[834903-43-4]
Formula:
C25H19N3O4
Target:
GPR55
Application Notes:
MCE Product type: Reference compound1
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