PROTAC PIN1 degrader-1 (compound D4) is a PROTAC targeting PIN1, with a DC50=1.8 nM. The GI50 of PROTAC PIN1 degrader-1 to MDA-MB-468 is >30 µM. PROTAC PIN1 degrader-1 is composed of target protein ligand PIN1 ligand-1 (HY-168038) (red part), E3 ligase ligand Thalidomide (HY-14658) (blue part), and PROTAC linker (black part)[1].
Molecular Weight:
917.02
CAS Number:
[3038591-59-9]
Formula:
C51H52N10O7
Target:
PIN1,PROTACs
Application Notes:
MCE Product type: Reference compound
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