CHI-KAT8i5 is a selective and orally active KAT8 inhibitor with a KD value of 19.72 µM. CHI-KAT8i5 does not bind to other proteins in HAT family (KAT2A, KAT2B, KAT5, and KAT7). CHI-KAT8i5 induces cancer cell apoptosis. CHI-KAT8i5 suppresses esophageal squamous cell carcinoma (ESCC) growth through targeting KAT8/c-Myc signaling pathway[1].
Molecular Weight:
523.69
Purity:
98.00
Formula:
C23H29N3O5S3
Target:
Apoptosis,Histone Acetyltransferase
Application Notes:
MCE Product type: Reference compound
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