MS-553 is a potent, ATP-competitive and reversible inhibitor of conventional PKC enzymes with Kis of 5.3 and 10.4 nM for human PKCbeta and PKCalpha, and IC50s of 2.3, 8.1, 7.6, 25.6, 57.5, 314, 808 nM for PKCalpha, PKCbetaI, PKCbetaII, PKCtheta, PKCgamma, PKC mu and PKCepsilon, respectively.
Molecular Weight:
500.61
Purity:
99.79
CAS Number:
[1046787-18-1]
Formula:
C25H37FN8O2
Target:
PKC
Application Notes:
MCE Product type: Reference compound
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