RK-851 is a highly selective and orally active delta-opioid receptor antagonist, with a negative logarithm of the antagonist concentration (pA2) of 8.84. TRK-851 exhibits the selectivity for the delta receptor of more than 100 times higher than that for the µ or kappa receptors. TRK-851 exhibits a potent antitussive effect in a rat model of capsaicin-induced cough. TRK-851 can be used for research on antitussive effects[1].
Molecular Weight:
472.55
CAS Number:
[189015-24-5]
Formula:
C29H29FN2O3
Target:
Opioid Receptor
Application Notes:
MCE Product type: Reference compound
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