LSD1-IN-42 (Compound 7ae) is an orally active LSD1 inhibitor that potently inhibits LSD1 activity (IC50 = 0.08 µM). LSD1-IN-42 downregulates PD-L1 expression and enhances T cell-mediated tumor killing effects. LSD1-IN-42 demonstrates significant anti-gastric cancer activity by inhibiting tumor cell invasion and migration[1].
Molecular Weight:
505.93
Formula:
C22H20ClN3O7S
Target:
Histone Demethylase,PD-1/PD-L1
Application Notes:
MCE Product type: Reference compound
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