PDHK1-IN-3 (Compound 29) is a selective PDHK1 inhibitor with an IC50 of 0.028 µM against PDHK1 and an IC50 of 0.120 µM against PDHK2. PDHK1-IN-3 inhibits the activity of PDHK1 by forming a covalent bond with Lys299 in PDHK1. PDHK1-IN-3 can be used in the research of autoimmune diseases, inflammatory diseases, and cancer[1].
Molecular Weight:
445.44
Formula:
C21H17F2N3O4S
Target:
PDHK
Application Notes:
MCE Product type: Reference compound
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