EZH2-IN-23, CAS [[3095068-20-2]] Preis auf Anfrage

Product Overview

• Article Name: EZH2-IN-23, CAS [[3095068-20-2]] Preis auf Anfrage
• Biozol Catalog Number: MCE-HY-174372
• Supplier Catalog Number: HY-174372
• Alternative Catalog Number: MCE-HY-174372-1UNIT
• Manufacturer: MedchemExpress
• Category: Biochemikalien

Product Description

EZH2-IN-23 (Compound 25) is an EZH2 inhibitor that exhibits potent enzymatic inhibition of the PRC2 complex (EZH2, EED, SUZ12, AEBP2, RbAp48) with a biochemical IC50 of 0.8 nM. EZH2-IN-23 inhibits H3K27 trimethylation in cellular assays, showing an IC50 of 40 nM. EZH2-IN-23 displays good rat PKproperties with 100 % oral bioavailability[1].

Product Properties

• Molecular Weight: 539.13
• CAS Number: [3095068-20-2]
• Formula: C29H35ClN4O2S
• Target: Histone Methyltransferase

Application Notes

• Application Notes: MCE Product type: Reference compound