Cenerimod (ACT-334441) is a potent, selective and orally active S1P1 receptor modulator, with an EC50 of 1 nM. Cenerimod shows more than 36 fold selctivity for hS1P1 over hS1P2, hS1P3, hS1P4, and hS1P5 receptor subtypes (EC50s=>10000, 228, 2134, and 36 nM, respectively). Cenerimod can attenuate murine experimental autoimmune encephalomyelitis (EAE) and murine sclerodermatous[1][2].
Molecular Weight:
453.53
Purity:
99.43
CAS Number:
[1262414-04-9]
Formula:
C25H31N3O5
Target:
LPL Receptor
Application Notes:
MCE Product type: Reference compound
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