ER degrader 12, CAS [[2376991-14-7]] Preis auf Anfrage

Catalog Number: MCE-HY-176955
Article Name: ER degrader 12, CAS [[2376991-14-7]] Preis auf Anfrage
Biozol Catalog Number: MCE-HY-176955
Supplier Catalog Number: HY-176955
Alternative Catalog Number: MCE-HY-176955-1UNIT
Manufacturer: MedchemExpress
Category: Biochemikalien
ER degrader 12 (Example 1) is an estrogen receptor (ER) degrader with IC50 values for ERalpha and ERbeta of 2.3 and 80.2 nM respectively (TR-FRET experiment). ER degrader 12 inhibits the proliferation of MCF-7 cells, with an IC50 of 1.53 nM. ER degrader 12 can be used for research on breast cancer[1].
Molecular Weight: 487.56
CAS Number: [2376991-14-7]
Formula: C26H32F3N5O
Target: Estrogen Receptor/ERR
Application Notes: MCE Product type: Reference compound