KAT6A/KAT7-IN-1 (Example 113) is a KAT6A and KAT7 inhibitor. The IC50 of KAT6A/KAT7-IN-1 for KAT6A is > 1 nM but 10 nM, while the IC50 for KAT7 is 1 nM. KAT6A/KAT7-IN-1 can inhibit the acetylation of H3K14 and H3K23. KAT6A/KAT7-IN-1 also inhibits tumor cell proliferation, with an IC50 of > 2 µM but 5 µM for CAMA-1. KAT6A/KAT7-IN-1 can be used in the study of cancer[1].
Molecular Weight:
495.55
Formula:
C25H25N3O6S
Target:
Histone Acetyltransferase
Application Notes:
MCE Product type: Reference compound
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