GSTO1-IN-4 is a selective, potent GSTO1-1 inhibitor (IC50 = 0.04 µM, KI = 0.16 µM). GSTO1-IN-4 shows low inhibition to GSTO2-2, GSTA1-1 and GSTP1-1. GSTO1-IN-4 shows a capacity to attenuate inflammation in mice and to significantly enhance the cytotoxicity of Cisplatin (HY-17394). GSTO1-IN-4 can be used for the study of inflammation and breast cancer[1].
Molecular Weight:
279.80
CAS Number:
[158890-33-6]
Formula:
C16H22ClNO
Target:
Glutathione S-transferase
Application Notes:
MCE Product type: Reference compound
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