SERT/5-HT-IN-1 is an orally active and potent dual target inhibitor of SERT/5-HT3A (SERT IC50 = 1.5 nM, NET IC50 = 49 nM, DAT IC50 = 91 nM, 5-HT3A Ki = 12 nM). SERT/5-HT-IN-1 has an IC50 of 39 nM to 5-HT3A. SERT/5-HT-IN-1 has a lower risk of liver, kidney, and cardiac toxicity. SERT/5-HT-IN-1 can be used for research on depressive disorders[1].
Molecular Weight:
258.38
Formula:
C15H18N2S
Target:
5-HT Receptor,Serotonin Transporter
Application Notes:
MCE Product type: Reference compound
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