AR ligand-49 (Compound 4q) is a dual ligand for the adenosine A2A receptor (A2AAR) and the A3 receptor (A3AR). Its Ki values are 15 and 4.5 nM respectively. AR ligand-49 exhibits reverse agonistic activity at hA2AAR and antagonistic activity at hA3AR. AR ligand-49 can be used for the study of the design and development of adenosine receptor ligands[1].
Molecular Weight:
429.50
Formula:
C19H23N7O3S
Target:
Androgen Receptor
Application Notes:
MCE Product type: Reference compound
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