GRL-03022 is a potent, selective and non-covalent G protein-coupled receptor kinase 5 (GRK5) inhibitor with an IC50 of 60 nM. GRL-03022 exhibits >16000-fold selectivity over GRK2 (IC50 > 1000 µM). GRL-03022 can be used for heart failure and cancer research[1].
Molecular Weight:
500.59
Formula:
C29H32N4O4
Target:
G Protein-coupled Receptor Kinase (GRK)
Application Notes:
MCE Product type: Reference compound
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