ERG-IN-5 (Compound M1) is a metabolite of ERG-IN-4 (HY-180918), and it is a hERG potassium channel inhibitor with an IC50 of 1.5 µM. ERG-IN-5 is cytotoxic to MTAPdel HCT116 and its CC50 is 28 nM. ERG-IN-5 can be used for the study of colon cancer[1].
Molecular Weight:
483.45
CAS Number:
[3047675-62-4]
Formula:
C23H20F3N7O2
Target:
Drug Metabolite,Potassium Channel
Application Notes:
MCE Product type: Reference compound
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