INSP-0154 is a potent creatine kinase B (CKB)/creatine transporter (SLC6A8) inhibitor. INSP-0154 binds to the SLC6A8 occluded pocket, prevents creatine transport into cells, and protects SLC6A8 cysteine residue C144 from irreversible inactivation. INSP-0154 inhibits creatine uptake in mouse heart tissue. INSP-0154 can be used for the research of cancer[1].
Molecular Weight:
170.17
Formula:
C6H10N4O2
Target:
Amino acid Transporter
Application Notes:
MCE Product type: Reference compound
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