VT102 is a TEAD1 inhibitor with a human IC50 of 391 nM. VT102 inhibits auto-palmitoylation, attenuates YAP/TEAD1 interaction, reduces expression of TEAD target genes, and inhibits YAP-mediated luciferase reporter activity. VT102 exerts weak cell growth inhibitory activity in cancer cells. VT102 can be used for the research of cancer[1].
Molecular Weight:
470.39
CAS Number:
[1119382-90-9]
Formula:
C21H20BrN5OS
Target:
YAP
Application Notes:
MCE Product type: Reference compound1
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