RTICBM-74 is a blood-brain barrier-permeable, selective CB1 allosteric modulator with IC50 values of 23 nM (calcium mobilization assay) and 153 nM ([35S]GTPgammaS assay). RTICBM-74 inhibits CB1 receptor signaling. RTICBM-74 reduces alcohol intake in rats. RTICBM-74 can be used for the research of alcohol use disorder[1].
Molecular Weight:
340.78
CAS Number:
[2130881-32-0]
Formula:
C19H14ClFN2O
Target:
Cannabinoid Receptor
Application Notes:
MCE Product type: Reference compound1
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