N 0840 is a neutral antagonist of adenosine A1 receptor (A1AR), with a Ki value of 279 nM in rats and 1185 nM in humans. N 0840 modulates adenosine A1 receptor to increase forskolin-induced cyclic 3',5'-adenosine monophosphate production, with a GTP shift value close to 1. N 0840 can be used in studies of neuroprotection, cardiovascular/renal function[1].
Molecular Weight:
217.27
CAS Number:
[109292-91-3]
Formula:
C11H15N5
Target:
Adenosine Receptor
Application Notes:
MCE Product type: Reference compound1
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