HKC54 is a selective TRPV2 antagonist with an IC50 of 0.4 µM. HKC54 binds directly to TRPV2 and inhibits TRPV2-mediated calcium influx. HKC54 inhibits glioblastoma cell migration in vitro and breast cancer metastasis in vivo. HKC54 can be used for the research of breast cancer lung metastasis[1].
Molecular Weight:
344.36
Formula:
C18H20N2O5
Target:
Calcium Channel,TRP Channel
Application Notes:
MCE Product type: Reference compound
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