HEP-50768, CAS [[3036387-75-1]]

Product Overview

• Article Name: HEP-50768, CAS [[3036387-75-1]]
• Biozol Catalog Number: MCE-HY-183050
• Supplier Catalog Number: HY-183050
• Alternative Catalog Number: MCE-HY-183050-1MG, MCE-HY-183050-5MG, MCE-HY-183050-10MG, MCE-HY-183050-25MG
• Manufacturer: MedchemExpress
• Category: Biochemikalien

Product Description

HEP-50768 is an orally active and selective MRGPRX4 (hX4) antagonist. HEP-50768 suppresses basal and bile-acid-stimulated hX4 activity. HEP-50768 binds the receptors transmembrane pocket and induces extracellular loop rearrangements. HEP-50768 modulates GPCR microswitch motifs and reduces bile-acid-induced pruritic scratching behaviors. HEP-50768 can be used for the research of cholestatic pruritus[1].

Product Properties

• Molecular Weight: 350.27
• CAS Number: [3036387-75-1]
• Formula: C16H10F4N4O
• Target: Mas-related G-protein-coupled Receptor (MRGPR)

Application Notes

• Application Notes: MCE Product type: Reference compound