SR-14968 is a full, allosteric and non-competitive MOR agonist, with an EC50 of 88 nM for MOR in mouse brainstem. SR-14968 stabilizes MOR in a G protein signaling state that is resistant to washout but reversible by antagonists. SR-14968 induces respiratory depression in mice. SR-14968 can be used in pain-related research[1].
Molecular Weight:
469.20
CAS Number:
[2133455-40-8]
Formula:
C20H20BrCl2N3O
Target:
Opioid Receptor
Application Notes:
MCE Product type: Reference compound
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