RQ-00203078 is a highly selective, potent and orally active TRPM8 antagonist with IC50s of 5.3 nM and 8.3 nM for rat and human TRPM8 channels, respectively. RQ-00203078 shows little inhibitory action against TRPV1, TRPA1, TRPV4, or TRPM2 channels[1][2].
Molecular Weight:
554.85
Purity:
99.84
CAS Number:
[1254205-52-1]
Formula:
C21H13ClF6N2O5S
Target:
TRP Channel
Application Notes:
MCE Product type: Reference compound
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