TG4-155 is a potent, brain-permeant and selective EP2 receptor antagonist with a Ki of 9.9 nM[1][2]. TG4-155 shows low nanomolar antagonist activity against only EP2 and DP1[1]. TG4-155 has an EP2 Schild KB of 2.4 nM and displays 550-4750-fold selectivity for EP2 over EP1, EP3, EP4 and IP, but only 14-fold selectivity against the DP1 receptor[2].
Molecular Weight:
394.46
Purity:
99.91
CAS Number:
[1164462-05-8]
Formula:
C23H26N2O4
Target:
Prostaglandin Receptor
Application Notes:
MCE Product type: Reference compound
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