BRL-52656 is a blood-brain barrier (BBB)-penetrable KOR receptor agonist that exhibits a biphasic effect. At low doses, BRL-52656 decreases blood pressure, whereas high doses have the opposite effect in spontaneously hypertensive rats. Additionally, BRL-52656 induces water diuresis by inhibiting the secretion of vasopressin (AVP)[1][2].
Molecular Weight:
390.87
CAS Number:
[115642-84-7]
Formula:
C19H26ClF3N2O
Target:
Opioid Receptor
Application Notes:
MCE Product type: Reference compound1
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