UBP-282 is a potent, selective and competitive AMPA and kainate receptor antagonist. UBP-282 inhibits the fast component of the dorsal root-evoked ventral root potential (fDR-VRP) with an IC50 value of 10.3 µM. UBP-282 antagonizes kainate-induced depolarisations of dorsal roots with a pA2 value of 4.96[1][2].
Molecular Weight:
333.30
CAS Number:
[544697-47-4]
Formula:
C15H15N3O6
Target:
iGluR
Application Notes:
MCE Product type: Reference compound
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