GYKI-47261 dihydrochloride is a competitive, orally active, and selective AMPA receptor antagonist with an IC50 of 2.5 µM. GYKI-47261 has broad spectrum anticonvulsive activity and neuroprotective effects. GYKI-47261 dihydrochloride is also a potent inducer of CYP2E1[1][2].
Molecular Weight:
395.71
CAS Number:
[1217049-32-5]
Formula:
C18H17Cl3N4
Target:
Cytochrome P450,iGluR
Application Notes:
MCE Product type: Reference compound
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