JX06 is a potent, selective and covalent inhibitor of PDK. JX06 inhibits PDK1, PDK2 and PDK3 with IC50s of 49 nM, 101 nM, and 313 nM, respectively. JX06 inhibits PDK1 activity via covalently binding to a cysteine residue in an irreversible manner. JX06 shows significant antitumor activity[1].
Molecular Weight:
324.51
Purity:
99.78
CAS Number:
[729-46-4]
Formula:
C10H16N2O2S4
Target:
Apoptosis,PDHK
Application Notes:
Reference compound
* VAT and and shipping costs not included. Errors and price changes excepted
