Naldemedine, CAS [[916072-89-4]] Preis auf Anfrage
Biozol Catalog Number:
MCE-HY-19627
Supplier Catalog Number:
HY-19627
Alternative Catalog Number:
MCE-HY-19627-1UNIT
Manufacturer:
MedchemExpress
Category:
Biochemikalien
Alternative Names:
S-297995
Naldemedine (S-297995) is an orally active µ-opioid receptor antagonist (PAMORA)[1]. Naldemedine shows potent binding affinities (Ki=0.34, 0.43, 0.94 nM, respectively) and antagonist activities (IC50=25.57, 7.09, 16.1 nM, respectively) for recombinant human µ-, delta-, and kappa- opioid receptors[2]. Naldemedine can be used in opioid-induced constipation (OIC) research[2]. Naldemedine is predicted to bind to 3CLpro encoded by SARS-CoV2 genome[3].
Molecular Weight:
570.64
CAS Number:
[916072-89-4]
Formula:
C32H34N4O6
Target:
Opioid Receptor
Application Notes:
MCE Product type: Reference compound
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