Enciprazine is an orally active non-benzodiazepine anxiolytic. Enciprazine acts as an agonist of 5-HT1A receptor (5-HT1AR) and an antagonist of alpha1-adrenergic receptor (alpha1-adrenergic receptor) . Enciprazine induces drug-related electroencephalogram changes by reducing the average power of delta waves and theta waves, and increasing the average power of alpha waves and fast beta waves. Enciprazine exhibits anti-aggressive activity, with only weak sedative and ataxic effects. Enciprazine regulates plasma corticosterone levels and activates the hypothalamic-pituitary-adrenal axis. Enciprazine can be used in research related to anxiety disorders, generalized anxiety syndrome and psychosis[1][2][3].
Molecular Weight:
432.51
CAS Number:
[68576-86-3]
Formula:
C23H32N2O6
Target:
5-HT Receptor,Adrenergic Receptor
Application Notes:
MCE Product type: Reference compound1
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