JNJ-63533054 is a potent, selective and orally active GPR139 agonist with an EC50 of 16 nM for human GPR139 (hGPR139). JNJ-63533054 shows selective for GPR139 over other GPCRs, ion channels, and transporters. JNJ-63533054 can cross the blood-brain barrier (BBB)[1][2].
Molecular Weight:
316.78
Purity:
99.80
CAS Number:
[1802326-66-4]
Formula:
C17H17ClN2O2
Target:
GPR139
Application Notes:
MCE Product type: Reference compound
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