LY-466195 is a selective and competitive GLUK5 receptor antagonist. LY-466195 antagonizes Kainate-induced currents with an IC50 value of 0.045 µM in rat dorsal root ganglion neurons. In HEK293 cells transfected with GLUK5, GLUK2/GLUK5, or GLUK5/GLUK66 receptors, LY466195 produces IC50 values of 0.08 µM, 0.34 µM, and 0.07 µM, respectively[1].
Molecular Weight:
346.37
CAS Number:
[317844-33-0]
Formula:
C16H24F2N2O4
Target:
iGluR
Application Notes:
MCE Product type: Reference compound
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