Tianeptine-d12, CAS [[1189870-26-5]] Preis auf Anfrage
Biozol Catalog Number:
MCE-HY-90003S
Supplier Catalog Number:
HY-90003S
Alternative Catalog Number:
MCE-HY-90003S-5MG,MCE-HY-90003S-500UG
Manufacturer:
MedchemExpress
Category:
Biochemikalien
Tianeptine-d12 is a deuterated analog of Tianeptine (HY-90003).Tianeptine is an atypical antidepressant. Tianeptine is a moderate-intensity agonist of the µ-opioid receptor (MOR), and to a lesser extent, is an agonist of the delta-opioid receptor (DOR). Tianeptine is a glutamate modulator that can enhance AMPA receptor and antagonize NMDA receptor. Tianeptine increases sensitivity of the alpha1 adrenergic receptor, which only manifests in chronic treatment. Tianeptine exerts neuroprotective effects under stress/inflammation-induced conditions, exhibiting anti-inflammatory and antioxidant properties. Tianeptine inhibits MMP-9 by suppressing the PI3K/Akt-mediated NF-kappaB pathway. Tianeptine can be used to alleviate symptoms of depression and anxiety, but does not cause sedative effects.
