Dienogest-13C,15N,d4 (STS 557-13C,15N,d4) is the 13C, 15N and deuterium labeled isotope of Dienogest (HY-B0084). Dienogest (STS-557) is an orally active and selective progesterone receptor agonist that effectively reduces the gene expression of COX-2, mPGES-1 and aromatase. Dienogest also inhibits the mRNA and protein expression of PGE2 synthase and the activation of NF-kappaB. Dienogest can be used in studies of endometriosis, menopause and menorrhagia[1][2].
Molecular Weight:
317.43
Formula:
C19 13CH21D4 15NO2
Target:
Isotope-Labeled Compounds,Progesterone Receptor
Application Notes:
MCE Product type: Isotope-Labeled Compounds
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