Cyclosporine A acetate-d4, Ciclosporin A acetate-d4, CsA acetate-d4
Cyclosporin A acetate-d4 (Cyclosporine A acetate-d4, Ciclosporin A acetate-d4) is a deuterium labeled Cyclosporin A (HY-B0579)[1]. Cyclosporin A (Cyclosporine A) is an immunosuppressant which binds to the cyclophilin and inhibits phosphatase activity of protein phosphatase 2B (PP2B/calcineurin) with an IC50 of 5 nM[2]. Cyclosporin A also inhibits CD11a/CD18 adhesion[3].