Crotamiton is a TRPV4 inhibitor. Crotamiton inhibits TRPV4 currents. Crotamiton inhibits TRPV4 selective agonist-induced pruritus-related behaviors in mice. Crotamiton inhibits Histamine- and Chloroquine-induced calcium influx via the H1R/TRPV1, MRGPRA3/TRPA1 pathways, and also suppresses calcium influx in primary mouse dorsal root ganglion neurons. Crotamiton is applicable to research related to pruritus, scabies, and non-scabietic pruritus[1][2].
Molecular Weight:
203.28
Purity:
98.07
CAS Number:
[483-63-6]
Formula:
C13H17NO
Target:
Parasite,TRP Channel
Application Notes:
MCE Product type: Reference compound
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