Hemicholinium 3 is a competitive inhibitor of the high affinity choline transporter (HACU) with a Ki value of 25 nM. Hemicholinium 3, a neuromuscular blocking agent which inhibits the synthesis and the release of acetylcholine (ACh)[1]. Hemicholinium 3 inhibits the Epibatidine-evoked contraction and [3H]acetylcholine release with IC50s of 897 nM and 693 nM, respectively[2].
Molecular Weight:
574.35
Purity:
99.86
CAS Number:
[312-45-8]
Formula:
C24H34Br2N2O4
Target:
Cholinesterase (ChE)
Application Notes:
MCE Product type: Reference compound
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