Gambogenic acid is an active ingredient that can be isolated from gamboge. Gambogenic acid acts as an effective inhibitor of EZH2, specifically and covalently binds to Cys668 within the EZH2-SET domain, and induces EZH2 ubiquitination. Gambogenic acid can be used for the research of cancer[1][2].
Molecular Weight:
630.77
Purity:
99.91
CAS Number:
[173932-75-7]
Formula:
C38H46O8
Target:
Histone Methyltransferase
Application Notes:
MCE Product type: Natural Products
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