CS-VIP 8 (hydrochloride)

Catalog Number: MCE-HY-P10948A
Article Name: CS-VIP 8 (hydrochloride)
Biozol Catalog Number: MCE-HY-P10948A
Supplier Catalog Number: HY-P10948A
Alternative Catalog Number: MCE-HY-P10948A-5MG,MCE-HY-P10948A-500UG,MCE-HY-P10948A-10MG,MCE-HY-P10948A-1MG
Manufacturer: MedchemExpress
Category: Proteine/Peptide
CS-VIP 8 hydrochloride is a selective allosteric WDR5 protein inhibitor (Ki= 0.008 µM). CS-VIP 8 hydrochloride induces conformational changes in the MLL1 complex, leading to the dissociation of MLL1 from the complex, inhibiting MLL1 histone methyltransferase activity and regulating HOX gene expression. CS-VIP 8 hydrochloride is promising for research of hematological diseases such as leukemia[1].
Molecular Weight: 961.40
Purity: 96.04
Formula: C43H53ClF4N12O7
Target: Histone Methyltransferase,WDR5
Application Notes: MCE Product type: Peptides