ELA-21 (human) is an apelin receptor agonist with a pKi of 8.52. ELA-21 (human) completely inhibits Forskolin-induced cAMP production and stimulates beta-arrestin recruitment with subnanomolar potencies. ELA-21 (human) is an agonist in G-protein-dependent and -independent pathways[1].
Molecular Weight:
2587.11
Purity:
99.97
CAS Number:
[2245073-05-4]
Formula:
C112H184N40O25S3
Target:
Apelin Receptor (APJ),Arrestin
Application Notes:
MCE Product type: Peptides
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