(EC50=3 nM). hMC1R agonist 1 shows at least 300-fold selectivity for hMC1R over hMC3R (b>EC50=902 nM), hMC4R (b>EC50=915 nM), and hMC5R (b>EC50=>1000 nM). hMC1R agonist 1 has the potential for the therapeutic intervention of melanocortin family[1].
Molecular Weight:
1107.35
Purity:
99.37
CAS Number:
[3028881-87-7]
Formula:
C54H70N14O8S2
Target:
Melanocortin Receptor
Application Notes:
MCE Product type: Reference compound1
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