RSK2-IN-4 (Compound 10) is a RSK2 inhibitor, with an inhibition rate of 13.73% on RSK2 activity at 10 µM. RSK2-IN-4 binds to the ATP-binding site of RSK2 in the NTKD (N-terminal kinase domain), with the electron-donating group at the 4-position of the phenyl ring being the key determinant for its inhibitory activity [1].
Molecular Weight:
258.71
CAS Number:
[62001-32-5]
Formula:
C13H11ClN4
Target:
Ribosomal S6 Kinase (RSK)
Application Notes:
MCE Product type: Reference compound
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