ALT-2074 (BXT-51071) is an orally active catalytic analogue of glutathione peroxidase. ALT-2074 is an inhibitor of human CYP3A, with its IC50 value ranging from 2.0 to 2.6 µM. ALT-2074 shows only a weak inhibitory effect on CYP3A in vivo, suggesting that it may not significantly affect the metabolism of CYP3A substrate drugs. ALT-2074 can be used to study inflammatory diseases characterized by reactive oxygen species, such as acute coronary syndrome[1].
Molecular Weight:
226.18
CAS Number:
[173026-17-0]
Formula:
C10H13NSe
Target:
Cytochrome P450,Glutathione Peroxidase
Application Notes:
MCE Product type: Reference compound
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