L-803087 is a potent and selective agonist of the growth inhibitor sst4 receptor with a Ki value of 0.7 nM for sst4, demonstrating over 280-fold selectivity compared to other growth inhibitory receptors. L-803087 induces AMPA-mediated synaptic responses in the hippocampus in vitro and increases seizures in alginate-induced seizure-busting mice in vivo.
Molecular Weight:
485.53
Purity:
97.58%
CAS Number:
[217480-26-7]
Formula:
C25H29F2N5O3
Target:
Somatostatin
T11800
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